Anti-Cancer Drug Discovery Using Synthetic Lethal Chemogenetic (SLC) Analysis

Abstract

I am developing a novel cell-based small-molecule screening approach that can identify inhibitors of any non-essential protein function through a surrogate synthetic lethal phenotype in the baker's yeast, Saccharomyces cerevisiae. Synthetic lethality (SL) is a form of genetic enhancement in which two mutations are lethal in combination, but the corresponding individual mutants are viable. Thus, a sensitized yeast strain carrying a mutation that is synthetic lethal with a gene of interest will be inviable in the presence of a chemical inhibitor of the target protein.

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Document Details

Document Type
Technical Report
Publication Date
Jul 01, 2004
Accession Number
ADA434327

Entities

People

  • David S. Bellows

Organizations

  • Mount Sinai Hospital, Toronto

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Abstracts
  • Cells
  • Drug Resistance
  • Genes
  • Genetic Enhancement
  • Genetic Phenomena
  • Genetics
  • Genome
  • Hospitals
  • Inhibition
  • Inhibitors
  • Lethality
  • Molecules
  • Neoplasms
  • Phenotypes
  • Platforms
  • Small Molecules

Fields of Study

  • Biology

Readers

  • Molecular Genetics

Technology Areas

  • Biotechnology
  • Biotechnology - Cancer Biotech