Cyclopentadienyl Rhenium (Technetium) Tricarbonyl Complexes Integrated in Estrogen Receptor Ligands for ER+ Tumor Imaging

Abstract

A class of breast tumors, known as ER+, contains significant concentrations of ER which functions to regulate cell growth, and mediate the action of estrogen antagonists. There is a need for the development non-invasive and reliable methods for the determination of tumor ER concentration in the identification of patients predicted to respond to hormone therapy. It has been shown that tumor ER concentration can be determined by imaging, using 18F-labeled ER selective ligands, and that the ER concentrations determined by imaging correlate well with those determined by immunoassay methods on surgical biopsies.

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Document Details

Document Type
Technical Report
Publication Date
Oct 01, 2004
Accession Number
ADA434829

Entities

People

  • John Katzenellenbogen
  • Nathan C. Ackroyd

Organizations

  • University of Illinois Urbana–Champaign

Tags

DTIC Thesaurus Topics

  • Alcohols
  • Alkenes
  • Alkynes
  • Biomedical Research
  • Breast Cancer
  • Chemical Synthesis
  • Chemistry
  • Chemotherapy
  • Controlled Atmospheres
  • Health Services
  • Illinois
  • Neoplasms
  • Organic Chemistry
  • Technetium
  • Therapy
  • Transition Metals
  • Universities

Fields of Study

  • Chemistry

Readers

  • Materials Science and Engineering.
  • Molecular and Cellular Biochemistry
  • Oncology and Biomarker-Based Cancer Detection.