An Activity-Dependent Assay for Ricin and Related RNA N-Glycosidases Based on Electrochemiluminescence

Abstract

Synthetic biotinylated RNA substrates were cleaved by the combined actions of ricin holotoxin and a chemical agent, N,N'-dimethylethylenediamine. The annealing of the product with a ruthenylated oligodeoxynucleotide resulted in the capture of ruthenium chelate onto magnetic beads, enabling the electrochemiluminescence (ECL)-based detection of RNA N-glycosidase activities of toxins. ECL immunoassays and the activity assay exhibited similar limits of detection just below signals with 0.1ng/ml of ricin; the ECL response was linear as the ricin concentration increased by two orders of magnitude. Activities were detected with other adenine-specific RNA N-glycosidases, including Ricinus communis agglutinin (RCA), saporin, and abrin II. The substrate that provided the greatest sensitivity was composed of a four-residue loop, GdAGA, in a hairpin structure. When the 2'-deoxyadenosine (dA) was substituted with adenosine (A), 2'-deoxyinosine, or 2'-deoxyuridine, toxin-dependent signals were abolished. Placing the GdAGA motif in a six-residue loop or replacing it with GdAdGA or GdAAA resulted in measurable activities and signal patterns that were reproducible for a given toxin. Data indicated that saporin and abrin II shared one pattern, while ricin and RCA shared a distinct pattern. A monoclonal antibody that enhanced the activities of ricin, RCA, and abrin II to different extents, thus improving the diagnostic potential of the assay, was identified.

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Document Details

Document Type
Technical Report
Publication Date
Jan 01, 2006
Accession Number
ADA456993

Entities

People

  • Charles C. Young
  • Mark A. Poli
  • Victor R. Rivera
  • William K. Keener

Organizations

  • United States Army Medical Research Institute of Infectious Diseases

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Adenine
  • Agglutinins
  • Antibodies
  • Biochemistry
  • Cells
  • Chemical Synthesis
  • Chemical Warfare Agents
  • Chemistry
  • Detection
  • Glycosidases
  • Immunoassay
  • Liquid Chromatography
  • Materials
  • Molecules
  • Organelles
  • Proteins
  • Ribonucleic Acids

Fields of Study

  • Biology
  • Chemistry

Readers

  • Data Mining and Knowledge Discovery.
  • Molecular Genetics
  • Molecular and Cellular Biochemistry