The Regulation of Nuclear Receptor Coactivator SRC-3 Activity Through Membrane Receptor Mediated Signaling Pathways

Abstract

SRC-3 interacts with steroid receptors in a ligand-dependent manner to activate receptor mediated transcription. A number of signaling pathways initiated by growth factors and hormones induce phosphorylation of SRC-3, regulating its function and contributing to its oncogenic potential. However, the range of mechanisms by which phosphorylation affects coactivator function remains largely undefined. We demonstrate here that the peptidyl-prolyl isomerase 1 (Pin1), which catalyzes the isomerization of phosphorylated Ser/Thr-Pro peptide bonds to induce conformational changes of its target proteins, interacts selectively and specifically with phosphorylated SRC-3. In addition, Pin1 and SRC-3 activate nuclear receptor regulated transcription synergistically. We present evidence that Pin1 modulates interactions between SRC-3 and CBP/p300. Depletion of Pin1 in NCF-7 human breast cancer cells reduces endogenous estrogen-dependent recruitment of p300 to the promoters of estrogen receptor-dependent genes. Our results suggest that Pin1 functions as a transcriptional coactivator of nuclear receptors by modulating SRC-3 coactivator protein-protein complex formation, and ultimately, by regulating the turnover of the activated SRC-3 oncoprotein.

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Document Details

Document Type
Technical Report
Publication Date
May 01, 2005
Accession Number
ADA460836

Entities

People

  • Ping Yi

Organizations

  • Baylor College of Medicine

Tags

DTIC Thesaurus Topics

  • Biomolecules
  • Breast Cancer
  • Chemical Compounds
  • Estrogens
  • Growth Factors
  • Hormones
  • Isomerases
  • Isomerization
  • Membranes
  • Neoplasms
  • Phosphorylation
  • Regulations

Fields of Study

  • Biology
  • Chemistry

Readers

  • Breast cancer cell signaling and growth regulation.
  • Molecular Biology and Genetics