Inhibition of Androgen-Independent Growth of Prostate Cancer by siRNA-Mediated Androgen Receptor Gene Silencing

Abstract

In current period, We first used a signal intra-tumoral injection of different amount of AAV particles to define a proper dosage for efficient virus distribution and knockdown of AR expression. The defined dose was 5.0 x 10^6 AAV particles per 100 mm^3 of tumor volume. Next, we used this dose to treat prostate cancer xenografts. We found that intra-tumoral injection of the ARHP8 but not GFP AAVs abolished tumor growth in LNCaP- and C4-2-derived xenografts in both castrated and shamoperated mice. Immunostaining results confirmed that the AR expression was dramatically down-regulated in AAV.ARHP8-injected tumors. In addition, a significant increase of apoptosis index (TUNEL assay) and dramatic decrease of proliferation index (BrdU incorporation assay) were found in AAV.ARHP8-injected tumors compared to the GFP control. These results demonstrated that the AR is critical for androgen-dependent survival and tumor growth in prostate cancer. Next year, we will repeat these experiments using two more prostate cancer cell line-derived xenografts.

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Document Details

Document Type
Technical Report
Publication Date
Feb 01, 2006
Accession Number
ADA462862

Entities

People

  • Benyi Li

Organizations

  • University of Kansas Medical Center

Tags

DTIC Thesaurus Topics

  • Androgen Receptors
  • Antisense Elements (Genetics)
  • Blood
  • Cell Line
  • Cell Physiological Processes
  • Cells
  • Chemistry
  • Epithelial Cells
  • Gene Expression
  • Genetics
  • Membrane Potentials
  • Neoplasms
  • Oncology
  • Programmed Cell Death
  • Prostate Cancer
  • Proteins
  • Therapy

Fields of Study

  • Biology

Readers

  • Aerosol Science/Aerosol Physics
  • Immunology
  • Prostate Cancer Biology.