Silica-Immobilized Enzymes for Multi-Step Synthesis in Microfluidic Devices (Postprint)
Abstract
The microfluidic combinatorial synthesis of 2-aminophenoxazin-3-one (APO) is reported. Individual microfluidic chips containing metallic zinc, silica-immobilized hydroxylaminobenzene mutase and silica-immobilized soybean peroxidase are connected in series to create a chem-enzymatic system for synthesis. Zinc catalyzes the initial reduction of nitrobenzene to hydroxylaminobenzene which undergoes a biocatalytic conversion to 2-aminophenol, followed by enzymatic polymerization to 2-aminophenoxazin-3-one. Silica-immobilization of enzymes allows the rapid stabilization and integration of a biocatalyst within a microfluidic device with minimal preparation. The system proved suitable for synthesis of a complex natural product (APO) from a simple substrate (nitrobenzene) under continuous flow conditions.
Document Details
- Document Type
- Technical Report
- Publication Date
- Oct 01, 2007
- Accession Number
- ADA481472
Entities
People
- Bosung S. Ku
- Heather R. Luckarift
- Jim C. Spain
- Jonathan S. Dordick
Organizations
- Air Force Research Laboratory