Potentiation of Prostate Cancer Radiotherapy Using Antiangiogenic and Antitumor Therapies

Abstract

Various antiangiogenic strategies have proven effective in preclinical tumor models, either as single agents or combined with radiation (RT). The current work aimed to evaluate whether treatment sequencing critically impacts tumor pathophysiological and therapeutic response. Using human prostate tumor models, axitinib, an inhibitor of VEGF receptors, was administered either before or after each daily RT fraction, and pathophysiological changes were monitored. Tumor growth inhibition was equivalent following the two combination schedules. Similar reductions in blood vessel counts were observed with each, tumor hypoxia increased, and pericytes progressively dissociated. These studies illustrate a clear advantage to combining axitinib with fractionated therapy, but argue against an acute radiosensitization or radioprotection of either the tumor cells or tumor vasculature. Instead, post- and pre-RT drug administration serve equally well in supplementing radiotherapeutic response.

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Document Details

Document Type
Technical Report
Publication Date
Oct 01, 2008
Accession Number
ADA504477

Entities

People

  • Bruce M. Fenton

Organizations

  • University of Rochester

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Alkenes
  • Basements
  • Biomedical Research
  • Blood
  • Blood Vessels
  • Cells (Biology)
  • Combination Therapy
  • Endothelial Cells
  • Growth Factors
  • Inhibition
  • Inhibitors
  • Medical Personnel
  • Membranes
  • Neoplasms
  • Prostate
  • Prostate Cancer
  • Therapy

Fields of Study

  • Biology
  • Medicine

Readers

  • Oncology (Cancer Research).
  • Systems Analysis and Design