A Mouse Model for in Vivo Detection and Disruption of TGF-Beta Signaling in Breast Cancer Metastasis

Abstract

Although the transforming growth factor-beta (TGF-beta) pathway has been implicated in breast cancer metastasis, its in vivo dynamics and temporal-spatial involvement in organ-specific metastasis have not been investigated. Here we engineered a xenograft model system with a conditional control of the TGF-beta-SMAD signaling pathway and a dual-luciferase reporter system for tracing both metastatic burden and TGF-beta signaling activity in vivo. Strong TGF-beta signaling in osteolytic bone lesions is suppressed directly by genetic and pharmacological disruption of the TGF-beta-SMAD pathway and indirectly by inhibition of osteoclast function with bisphosphonates. Notably, disruption of TGF-beta signaling early in metastasis can substantially reduce metastasis burden but becomes less effective when bone lesions are well established. Our in vivo system for real-time manipulation and detection of TGF-beta signaling provides a proof of principle for using similar strategies to analyze the in vivo dynamics of other metastasisassociated signaling pathways and will expedite the development and characterization of therapeutic agents.

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Document Details

Document Type
Technical Report
Publication Date
Sep 01, 2009
Accession Number
ADA512330

Entities

People

  • Manav Korpal

Organizations

  • Princeton University

Tags

DTIC Thesaurus Topics

  • Antineoplastic Agents
  • Biological Sciences
  • Body Weight
  • Bone And Bones
  • Bone Diseases
  • Breast Cancer
  • Cell Line
  • Cells
  • Chemistry
  • Detection
  • Growth Factors
  • Molecular Biology
  • Neoplasms
  • Peptide Growth Factors
  • Peptides
  • Proteins
  • Three Dimensional

Fields of Study

  • Biology

Readers

  • Oncology (Cancer Research).

Technology Areas

  • Biotechnology
  • Biotechnology - Cancer Biotech