A Role for MEK-Interacting Protein 1 in Hormone Responsiveness of ER Positive Breast Cancer Cells

Abstract

Our results have revealed a critical and previously unreported role for the small scaffold protein MP1 in the survival of ER-positive, but not ER-negative breast cancer cell lines. Blocking MP1 expression using siRNA leads to apoptotic cell death in ER-positive MCF-7, LCC9 and T47D cells, but not in ER-negative MDA-MB-231, SKBr3 and BT-549 cells. Overexpression of MP1 may also be toxic to ER-positive cells, since MCF-7 derivatives expressing ectopic MP1 are unstable and rapidly lose expression of the transfected MP1 gene upon passage. The mechanism by which MP1 affects survival of ER-positive breast cancer cells is not known, but may be the result of alterations in ER levels and/or functions. In support of this hypothesis, MP1 knockdown leads to decreased ER levels, and MP1 overexpression to increased ER levels. Together, out data strongly suggest that MP1 could provide a novel target for the treatment of ER-positive breast tumors. Future experiments will investigate the mechanism(s) by which MP1 regulates survival of ER-positive breast cancer cells, and those by which it regulates ER levels and function.

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Document Details

Document Type
Technical Report
Publication Date
Jul 01, 2009
Accession Number
ADA514031

Entities

People

  • Susan E. Conrad

Organizations

  • Michigan State University

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Antibodies
  • Apoptosis
  • Azo Compounds
  • Biomedical Research
  • Breast Cancer
  • Cell Line
  • Cell Physiological Processes
  • Cells
  • Estrogens
  • Gene Expression
  • Genes
  • Genetics
  • Inhibition
  • Medical Personnel
  • Neoplasms
  • Survival
  • Tumor Cell Line

Fields of Study

  • Biology

Readers

  • Breast cancer cell signaling and growth regulation.
  • Military/Explosive Ordnance Disposal (EOD) Technology
  • Molecular Biology and Genetics