Characterization of IKBKE as a Breast Cancer Oncogene

Abstract

Previous work in the Hahn Lab has identified IKBKE as a novel breast cancer oncogene that is capable of human mammary cell transformation. Amplification and overexpression of IKKepsilon was observed in a significant percentage of human breast cancer cell lines and primary tumor samples. Additionally, breast cancer cell lines carrying the IKBKE amplicon showed decreased viability in response to IKKepsilon suppression by shRNA. Our work has also demonstrated that IKKepsilon is a non-canonical IKK (IkappaB kinase) family member that activates the NF-kappaB pathway and that this activity is essential for cell transformation. However, it is known that IKKepsilon not does participate in the canonical IKK complex to activate NF-kappaB signaling. Though recent work has sought to identify the downstream targets of IKKepsilon, the mechanism of its upstream regulation is not well-understood. Thus, I propose to further our understanding of IKKepsilon function by investigating the upstream regulation of IKKepsilon - specifically, the role of ubiquitination in IKKepsilon-mediated cell transformation. In addition, I am to investigate the role of IKKepsilon in breast cancer initiation and maintenance in vivo through the generation of a constitutive and an inducible transgenic mouse model.

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Document Details

Document Type
Technical Report
Publication Date
Oct 01, 2009
Accession Number
ADA515797

Entities

People

  • Alicia Zhou

Organizations

  • Dana–Farber Cancer Institute

Tags

DTIC Thesaurus Topics

  • Amino Acids
  • Biomedical Research
  • Breast Cancer
  • Cell Line
  • Cells
  • Demographic Cohorts
  • Department Of Defense
  • Epithelial Cells
  • Glands
  • Maintenance
  • Mammary Glands
  • Mass Spectrometry
  • Neoplasms
  • Phenotypes
  • Proteins
  • Regulations
  • Spectrometry

Readers

  • Data Mining and Knowledge Discovery.
  • Molecular Biology and Genetics