Identification of Estrogen Receptor Beta Binding Sites in the Human Genomes

Abstract

ER knock-out mice developed prostatic hyperplasia at late age, suggesting an important role of ER in the development of the prostate as well as prostate cancer. Here we describe a study that thoroughly investigates the genomic function of ER . A FLAG-tagged ER was stably expressed in MCF7 C4-12 cells, which allowed ER transcriptional activity to be studied in an ER -independent background. Interestingly, in our chromatin immunoprecipitation followed by sequencing (ChIP-seq) analyses, looking at ER global binding sites, while the most prevalent binding motif was the canonical ERE, ~30% of ER binding regions also carried the binding motif of EBF1 (Early B-cell Factor 1). Further investigations revealed EBF1 downregulated ER protein stability and transcriptional activity via a direct interaction. These results, at least to our knowledge, are the first to indicate crosstalk between EBF and ER activities on a large scale. Moreover, in conjunction with global run-on followed by sequencing (GRO-seq), looking at nascent RNA generated at the time of ER binding events, still to be completed, our results should reveal a global picture of how ER regulates its direct target genes, as well as the role of EBF proteins in this process.

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Document Details

Document Type
Technical Report
Publication Date
Aug 01, 2011
Accession Number
ADA549088

Entities

People

  • Thien Le

Organizations

  • University of Chicago

Tags

DTIC Thesaurus Topics

  • Biomedical Research
  • Breast Cancer
  • Cancer
  • Cell Line
  • Cells
  • Chromosome Structures
  • Co-Channel Interference
  • Estrogens
  • Genetic Structures
  • Genome
  • Human Genome
  • Neoplasms
  • Prostate
  • Prostate Cancer
  • Proteins
  • Sex Hormones
  • Transcription Factors

Fields of Study

  • Biology

Readers

  • Breast cancer cell signaling and growth regulation.
  • Molecular Genetics
  • Molecular and genetic basis of cancer.