Molecular Innovations Towards Theranostics of Aggressive Prostate Cancer

Abstract

In this project, we propose to develop a new drug delivery vehicle based on dendrimer nanotechnology for personalized medicine. This new class of nanoplatforms contains imaging probe and molecular medicine with a cancer-specific targeting capability which is able to target cancer cells, monitor drug delivery and tumor response to achieve a see and treat strategy as a new concept of molecular medicine. Specifically, One Partner PI s lab will make dendrimers bearing functional handles to conjugate with chelating agents provided by the Initiating PI s lab for PET imaging and therapeutic peptides provided by another Partner PI s lab for the treatment of aggressive prostate cancer. In the 1st year, the Initiating PI s lab has designed and synthesized the proposed bifunctional chelator scaffold system, CB-TE2A(tBu)2-N3 for the further construction of dendrimer-based theranostic agents for aggressive prostate cancer. In the meanwhile, the design concept has been extended to synthesize a bivalent imaging probe for quantitative PET imaging of PSMA expression in prostate cancer.

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Document Details

Document Type
Technical Report
Publication Date
Sep 01, 2013
Accession Number
ADA590551

Entities

People

  • Xiankai Sun

Organizations

  • University of Texas at Dallas

Tags

DTIC Thesaurus Topics

  • Biomedical Research
  • Blood Proteins
  • Chelate Compounds
  • Chemical Compounds
  • Chemical Synthesis
  • Chemistry
  • Construction
  • Dendrimers
  • Molecules
  • Nanotechnology
  • Neoplasms
  • Personalized Medicine
  • Prostate
  • Prostate Cancer
  • Targeting
  • Targets
  • Theranostics

Readers

  • Medical Imaging.
  • Nanocomposite Materials Science
  • Oncology

Technology Areas

  • Biotechnology
  • Biotechnology - Cancer Biotech