Chemically Modified Bacteriophage as a Streamlined Approach to Noninvasive Breast Cancer Imaging

Abstract

I have been able to convert cell surface marker-specific phage identified from library screens into imaging agents that can target and differentiate breast cancer cell types. This is accomplished by using efficient synthetic protocols to conjugate small molecules to phage coat proteins. In the current work, I have examined the use of phage targeting HER2, EGFR, HER3, CD44, and CD73 as immunofluorescence agents in order to visualize these cell surface receptors in cell button models of cancer tissues. Furthermore, I have initiated work whereby the targeting moieties (single chain antibody fragments, or scFv s) displayed by the filamentous phage are displayed on significantly smaller phage types (nanophage), which can be modified similarly and may possess improved biodistribution characteristics compared with the full length fd. I have also initiated the study of chemically modified icosahedral bacteriophage MS2 in order to target specific breast cancer-associated cell surface receptors in cell culture and mouse models of cancer. The work described in this final report ended on July 30, 2013, because I accepted an independent academic position in the chemistry department at the University of Massachusetts, Amherst.

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Document Details

Document Type
Technical Report
Publication Date
Dec 01, 2013
Accession Number
ADA596735

Entities

People

  • Michelle E. Farkas

Organizations

  • University of California, Berkeley

Tags

DTIC Thesaurus Topics

  • Breast Cancer
  • Cell Physiological Processes
  • Chemical Synthesis
  • Chemistry
  • Culture Techniques
  • Detection
  • Detectors
  • Genetic Engineering
  • Leviviridae
  • Liquid Chromatography
  • Mass Spectrometry
  • Materials Science
  • Molecular Biology
  • Neoplasms
  • Proteins
  • United States
  • Viral Structures

Fields of Study

  • Biology

Readers

  • Molecular Biology and Genetics
  • Molecular and Cellular Biochemistry
  • Systems Analysis and Design