Extracellular Hsp90 as a Novel Epigenetic Regulator of EMT and Metastatic Risk in Prostate Cancer

Abstract

In general, the role of eHsp90 in tumor progression has not been well characterized Our work provides novel mechanistic insights into the EMT-promoting activity of eHsp90. Our preliminary findings indicate that eHsp90 is a newly identified regulator of the oncogenic polycomb regulator EZH2. eHsp90 was found to induce EZH2 expression and to direct its recruitment to the promoters of target genes. In this latter capacity, eHsp90 promoted EZH2 s methyltransferase activity, enabling the repression of tumor suppressor genes such as the EMT gatekeeper E-cadherin. Moreover, xenograft studies demonstrate that an eHsp90-EZH2 axis is essential for eHsp90-mediated tumor invasion. Therefore, our findings implicate an eHsp90-EZH2 oncogenic pathway that contributes to early invasive events in prostate cancer.

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Document Details

Document Type
Technical Report
Publication Date
Oct 01, 2013
Accession Number
ADA603247

Entities

People

  • Jennifer S. Isaacs

Organizations

  • Medical University of South Carolina

Tags

DTIC Thesaurus Topics

  • Biomedical Research
  • Cancer
  • Cell Line
  • Cell Movement
  • Cells
  • Department Of Defense
  • Diseases And Disorders
  • Inhibitors
  • Medical Personnel
  • Metastasis
  • Molecules
  • Neoplasms
  • Prostate
  • Prostate Cancer
  • Regulators
  • Small Molecules
  • Tissues

Fields of Study

  • Biology

Readers

  • Molecular Biology and Genetics