Molecular Innovations Toward Theranostics of Aggressive Prostate Cancer

Abstract

In this project, we propose to develop a new drug delivery vehicle based on dendrimer nanotechnology for personalized medicine. This new class of nanoplatforms contains imaging probe and molecular medicine with a cancer-specific targeting capability which is able to target cancer cells, monitor drug delivery and tumor response to achieve a see and treat strategy as a new concept of molecular medicine. Specifically, One Partner PI s lab will make dendrimers bearing functional handles to conjugate with chelating agents provided by the Initiating PI s lab for PET imaging and therapeutic peptides provided by another Partner PI s lab for the treatment of aggressive prostate cancer. In the 2nd year, the Initiating PI s lab has designed and synthesized three enantiopure chelator scaffolds for copper radiopharmaceuticals using a well-validated integrin v 3 ligand. In addition, a theranostic molecular drug conjugate (MDC) design was accomplished. Such design will be modified and incorporated into the dendrimeric platforms to accomplish further Aims in this project.

Open PDF

Document Details

Document Type
Technical Report
Publication Date
Sep 01, 2014
Accession Number
ADA612560

Entities

People

  • Xiankai Sun

Organizations

  • University of Texas at Dallas

Tags

DTIC Thesaurus Topics

  • Alkanes
  • Chelate Compounds
  • Chemical Compounds
  • Chemical Synthesis
  • Chemistry
  • Column Chromatography
  • Detectors
  • Glutamic Acid
  • Liquid Chromatography
  • Molecules
  • Neoplasms
  • Nuclear Medicine
  • Organic Chemistry
  • Prostate
  • Prostate Cancer
  • Radiopharmaceuticals
  • Therapy

Readers

  • Medical Imaging.
  • Nanocomposite Materials Science
  • Oncology (Cancer Research).

Technology Areas

  • Biotechnology
  • Biotechnology - Cancer Biotech