1,2-Dicyclopropylethyne and (Cyclopropylethynyl)cyclobutane from an Efficient Synthesis of 1,2-(omega-Haloalkyl)ethynes and 1-Cycloalkyl-2-(omega-haloalkyl)ethynes (Pre Print)
Abstract
Lithium acetylides, generated from terminal acetylenes with n-BuLi in THF at -70 degrees C, react chemoselectively with omega-haloalkyl tosylate in the presence of 10 mole % of Bu4NI at 70 degrees C to furnish omega-haloalkyl acetylenes in very good yields. The omega-haloalkyl acetylenes undergo intramolecular alkylation with LDA to provide dicycloalkyl-ethynes.
Document Details
- Document Type
- Technical Report
- Publication Date
- Feb 09, 2012
- Accession Number
- ADA613652
Entities
People
- Jacob C. Marcischak
- Suresh C. Suri
Organizations
- Air Force Research Laboratory