Toxicity Testing of Antimalarial Drugs in Swine. I. A Study of Quinine Sulfate Toxicity.

Abstract

Quinine sulfate administered orally to swine in doses of 361 mg/kg/day (milligrams/kilograms/day) resulted in an LD 100/10 (Lethal dose 100/10), whereas, 180 mg/kg/day produced death in one of four pigs in 30 days, and no ill effects were observed in animals that received 45 mg/kg/day for 30 days. The most consistent symptoms observed were: emesis, depression, ataxia, partial to complete loss of sight and convulsions. The hematologic and biochemical results were very unimpressive, with few changes. The significant gross lesions may be summarized as: a hemorrhagic disorder, corneal lesions and alopecia. The most significant microscopic lesions are vacuolization of neurons, corneal lesions, bone marrow lesions and degenerative lesions of the arteriolar walls. Keywords: U/A Reports, Toxicity, Antimalarial, Drugs, Swine, Testing, Pharmacology, Quinine sulfate, Medical research. (jg)

Document Details

Document Type
Technical Report
Publication Date
Jun 30, 1967
Accession Number
ADA955926

Entities

People

  • Chester A. Gleiser
  • Kenneth R. Pierce
  • Randolph S. Brown
  • Thomas W. Dukes
  • William W. Bay

Organizations

  • Texas A&M University

Tags

Communities of Interest

  • Biomedical

DTIC Thesaurus Topics

  • Addiction
  • Antimalarials
  • Bacterial Infections And Mycoses
  • Biomedical Research
  • Bone Marrow
  • Bones
  • Chemically-Induced Disorders
  • Depression
  • Diseases And Disorders
  • Drug Abuse
  • Hematologic Diseases
  • Lethal Dosage
  • Mental Disorders
  • Pharmacology
  • Skin Diseases
  • Toxicity

Fields of Study

  • Medicine

Readers

  • Cardiovascular Physiology
  • Parasitology and Pharmacology of Malaria.
  • Toxicology/Environmental Toxicology