Synthesis of Improved Antileishmanial and Antitrypanosomal Drugs Treatment and Prophylaxis

Abstract

The program is directed at the preparation of improved antileishmanial and antitrypanosomal drugs. During the past year 13 target compounds were submitted for testing against L. donovani, T. rhodesiense and T. cruzi. Two candidate antileishmanials are modified 8-aminoquinolines. Eleven compounds were directed primarily against T. cruzi. These included seven 2,2- di(or tri)aryldimethyl(or dihydro)aminomethylethylenes and four 1-amidoximino-2, 2-di(or tri)diarylethylenes.

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Document Details

Document Type
Technical Report
Publication Date
Nov 01, 1986
Accession Number
ADB110976

Entities

People

  • A. B. Ash
  • A. Markovac
  • C. L. Stevens
  • D. J. Dagli
  • G. S. Wu
  • R. L. Kalamas

Tags

DTIC Thesaurus Topics

  • Acetic Acid
  • Acids
  • Alcohols
  • Alkanes
  • Alkenes
  • Aluminum Hydride
  • Amines
  • Biomedical Research
  • Chlorides
  • Cold Water
  • Column Chromatography
  • Hydrochloric Acid
  • Ketones
  • Maleic Acid
  • Nitriles
  • Sodium Compounds
  • Sodium Hydroxide

Fields of Study

  • Chemistry
  • Medicine

Readers

  • Parasitology and Pharmacology of Malaria.