Acetylcholinesterase and Acetylcholine Receptor

Abstract

This research seeks information about the properties and amino acid content of the active site of acetylcholinesterase (AcChE). It is based largely on the view that the subsite at which the positively charged Beta-substituent of the natural substrate, acetylcholine (AcCh), binds is not anionic, as is generally accepted, but uncharged and complementary to the trimethyl substituted character of that substituent. The subsite would be more specifically explored by uncharged reagents, while positive reagents would react at peripheral negative sites. Thus, uncharged irreversible and reversible inhibitors and substrates are obtained or synthesized and their reactions with the enzyme are studied. Keywords: Torpedo nobiliana; Chromatography; Electrophoresis.

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Document Details

Document Type
Technical Report
Publication Date
Jan 21, 1985
Accession Number
ADB112772

Entities

People

  • Saul G. Cohen

Organizations

  • Brandeis University

Tags

Communities of Interest

  • Biomedical
  • Weapons Technologies

DTIC Thesaurus Topics

  • Acetic Acid
  • Alcohols
  • Alkenes
  • Animal Structures
  • Aromatic Compounds
  • Chemical Synthesis
  • Chemistry
  • Contracts
  • Electrophoresis
  • Ethers
  • Fish
  • Gel Electrophoresis
  • Hydrophobic Properties
  • Inhibition
  • Ketones
  • Organic Chemistry
  • Universities

Fields of Study

  • Biology
  • Chemistry

Readers

  • Analytical Chemistry
  • Neurotoxicology
  • Systems Analysis and Design