Novel Fatty Acid Lipoxygenases in the Development of Human and Murine Prostate Cancer

Abstract

Changes in arachidonic acid (AA) metabolism may be crucial in development or progression of prostate adenocarcinoma (Pca). By immunohistochemistry, western blots, Northern blots, and enzyme assays, we have detected the uniform expression of a novel lipoxygenase, 15-LOX-2, in benign prostate. 15-LOX-2 and 15-HETE formation are substantially reduced or lost in the vast majority of Pca. In contrast to uniform 15-LOX-2 immunostaining in benign glands, tumors were focally (>25 %) and completely 15- LOX-2 negative in 59/97 (61 %) and 41/97 (42 %), respectively. In paired tissues from the same patients, 15-HETE formation and 15-LOX-2 mRNA were reduced in tumor vs. benign in 12/14 and 10/11, respectively. In contrast, significant changes in 5-HETE and 12-HETE formation have not been detected. Increased COX-2 mRNA was detected in 3/7 tumors vs. benign. 15-HETE may be a ligand for peroxisome proliferator activated receptors (PPARs), particularly PPARgamma. By RT-PCR, we have detected mRNA for PPARalpha, beta, and gamma in 18/18 benign and in 9/9 tumor specimens. 15-HETE induced PPAR gamma- dependent transcription in Pca cell lines. 15-HETE/ PPAR gamma signaling effects on cell proliferation and differentiation are being examined.

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Document Details

Document Type
Technical Report
Publication Date
Oct 01, 1999
Accession Number
ADB258930

Entities

People

  • Scott Shappell

Organizations

  • Vanderbilt University

Tags

DTIC Thesaurus Topics

  • Antineoplastic Agents
  • Carcinoma
  • Cell Physiological Processes
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Enzyme Inhibitors
  • Health Services
  • Liquid Chromatography
  • Medical Personnel
  • Neoplasms
  • Oncology
  • Prostate Cancer

Fields of Study

  • Biology

Readers

  • Oncology and Biomarker-Based Cancer Detection.
  • Prostate Cancer Biology.