Development of a Monoclonal Antibody Against Estrogen Quinone-Adducted Proteins as Potential Biomarkers of Breast Cancer Risk

Abstract

The purpose of this research is to develop a Specific monoclonal antibody (MAb) for intracellular detection and quantification of E2-3,4-Q adducted to proteins, as a potential biomarker of breast cancer risk. An established, protein-coupling chemistry was applied successfully to production of an immunogen, via linkage of E2-3,4-Q to cationized protein, through a short linker. A coating complex for indirect ELISA and a low molecular-weight conjugate for competitive ELISA were prepared by spontaneous adduction of E2-3,4-Q to an unmodified protein and a short-chain molecule with a primary amino group respectively. ELISA screening identified a hybridoma producing relatively large amounts of MAb with high signal-to- noise ratio. The affinity constant (0.5 x 10(exp 8) M(exp -1) for binding to E2-3,4-Q was determined by competitive ELISA. In specifically designed immunohistochemical (IHC)-staining protocols, the antibody produced intense and specific staining with no detectable cross-reactivity to E2-2,3-Q and little or no background. Failure to detect IHC staining in paraffin sections of ACI rat breast-tumors or human breast tumors is associated with loss of the epitope during microwave recovery or formalin fixation. Optimization of tissue fixation is required for validation studies that can be based on Quantitative Fluorescence Imaging Analysis or Surfaced-Enhanced Laser Desorption Ionization/tandem mass spectrometry.

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Document Details

Document Type
Technical Report
Publication Date
Jun 01, 2002
Accession Number
ADB282748

Entities

People

  • George P. Casale

Organizations

  • University of Nebraska Medical Center

Tags

DTIC Thesaurus Topics

  • Albumins
  • Alcohols
  • Alkanes
  • Antibodies
  • Biological Markers
  • Biological Staining And Labeling
  • Breast Cancer
  • Cells
  • Chemical Synthesis
  • Chemistry
  • Macromolecules
  • Mass Spectrometry
  • Molecular Weight
  • Molecules
  • Neoplasms
  • Organic Chemistry
  • Proteins

Fields of Study

  • Biology

Readers

  • Molecular and Cellular Biochemistry
  • Oncology and Biomarker-Based Cancer Detection.

Technology Areas

  • Directed Energy