Alanine Scan of Endothelin,

Abstract

In Order to get an insight into the endothelin's (ET) structural requirements for vasoconstrictor activity, a series of analogs was synthesized by SPPS, using the Boc-benzyl protecting group strategy. The paper describes the L-alanine scan, in which each non-cysteinyl residue was substituted individually with Ala.

Document Details

Document Type
Technical Report
Publication Date
Jan 01, 1992
Accession Number
ADP008422

Entities

People

  • J. P. Tam
  • J. W. Zhang
  • M. Galantino
  • R. De Castiglione
  • Wenxin Liu

Organizations

  • The Rockefeller University

Tags

DTIC Thesaurus Topics

  • Alanine
  • Chemical Compounds
  • Chemical Synthesis
  • Chemistry
  • Massachusetts

Fields of Study

  • Chemistry

Readers

  • Cardiovascular Physiology
  • Molecular and Cellular Biochemistry
  • Systems Analysis and Design