A Melanotropic Peptide Induces Pigmentation (Tanning) of Human Skin,

Abstract

We have designed and biologically characterized an analog of alpha-melanocyte stimulating hormone with the following structure: Ac-Ser-Tyr-Ser-Nle-Glu-His-D-Phe-Arg-Trp-Gly-Lys-Pro-Val-NH2. The hormone analog is superpotent, prolonged acting and is resistant to inactivation by sera and proteolytic enzymes. This peptide stimulates various pigmentation in the mouse when administered topically or when injected subcutaneously. Following FDA and Human Subjects Committee approval, the peptide was delivered by subcutaneous injection to human volunteers in a phase-I clinical trial.

Document Details

Document Type
Technical Report
Publication Date
Jan 01, 1992
Accession Number
ADP008432

Entities

People

  • M. E. Hadley
  • N. Levine
  • R. T. Dorr
  • S. D. Sharma
  • V. J. Hruby

Organizations

  • University of Arizona

Tags

DTIC Thesaurus Topics

  • Anatomy
  • Biological Sciences
  • Cells (Biology)
  • Chemistry
  • Clinical Trials
  • Continents
  • Epithelial Cells
  • Geographic Regions
  • Massachusetts
  • Volunteers

Fields of Study

  • Biology

Readers

  • Molecular and Cellular Biochemistry
  • Prostate Cancer Biology.
  • Toxicology/Environmental Toxicology