A Series of Highly Selective Thrombin Inhibitors,

Abstract

Tripeptide aldehydes such as Boc-D-Phe-Pro-Arg-H exhibit potent direct inhibition of thrombin. We have evaluated the structural and conformational role of the amino acid residue in position one of Boc-D-Phe-Pro-Arg-H.

Document Details

Document Type
Technical Report
Publication Date
Jan 01, 1992
Accession Number
ADP008543

Entities

People

  • Charles S. Campbell
  • Donetta S. Gifford-moore
  • Gerald F. Smith
  • Robert B. Rothenberger
  • Robert T. Shuman

Tags

DTIC Thesaurus Topics

  • Aldehydes
  • Amino Acids
  • Blood Coagulation Factors
  • Chemical Compounds
  • Chemical Synthesis
  • Chemistry
  • Inhibition
  • Inhibitors
  • Massachusetts
  • Organic Chemistry

Fields of Study

  • Chemistry

Readers

  • Molecular and Cellular Biochemistry