Determination of Subpicogram Quantities of Drugs and Narcotics in Urine of Human Subjects.

Abstract

The urinary excretions of methaqualone and 6-hydroxymethaqualone (free and conjugated) were studied in a normal male subject over a period of 30 days using stable isotope dilution analysis and field ionization mass spectrometry. The terminal half-lives of three compounds were estimated to be about 70 hr. These results were tentatively interpreted in terms of a multicomponent pharmacokinetic model. The ability of isotope dilution analysis using field ionization mass spectrometry to detect minute quantities of drugs in urine was thoroughly evaluated by these experiments. The sensitivity limit was between 0.1 and 1 ng/ml of urine, and was primarily limited by the chemical purity of the isolated drug or metabolite. (Author)

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Document Details

Document Type
Technical Report
Publication Date
Apr 01, 1976
Accession Number
ADA039107

Entities

People

  • Henry D'a. Heck
  • James H. Mcreynolds
  • Michael Anbar

Organizations

  • SRI International

Tags

DTIC Thesaurus Topics

  • Albumins
  • Alcohols
  • Antidepressants
  • Blood Proteins
  • Cellular Structures
  • Chemical Reactions
  • Chemistry
  • Chromatography
  • Equations
  • Health Services
  • Ionization
  • Kinetics
  • Mass Spectra
  • Mass Spectrometry
  • Pharmacology
  • Spectra
  • Spectrometry

Fields of Study

  • Chemistry

Readers

  • Brain and Cognitive Science; Experimental Psychology; Cognitive Neuroscience
  • Solar Physics
  • Toxicology/Environmental Toxicology